I-Pharmacodynamics ceftiofur iyikilasi le-β -lactam lemithi elwa namagciwane, enesenzo esibanzi se-bactericidal, esisebenza ngempumelelo ngokumelene nama-bacteria e-gram-positive kanye negram-negative (kuhlanganise namagciwane akhiqiza i-β-lactamase). Indlela yayo ye-antibacterial iwukuvimbela ukwakheka kodonga lwamaseli e-bacterial futhi kuholele ekufeni kwamabhaktheriya. Amagciwane azwelayo ikakhulukazi i-pasteurella multiplex, i-pasteurella hemolyticus, i-actinobacillus pleuropneumoniae, i-salmonella, i-escherichia coli, i-streptococcus, i-staphylococcus, njll. Amanye ama-pseudomonas aeruginosa, ukumelana ne-enterococcus. Umsebenzi we-antibacterial walo mkhiqizo unamandla kune-ampicillin, futhi umsebenzi omelene ne-streptococcus unamandla kune-fluoroquinolones.
I-Pharmacokinetics ceftiofur imuncwa ngokushesha nangokubanzi ngemijovo ye-intramuscular and subcutaneous, kodwa ayikwazi ukweqa umgoqo wobuchopho begazi. Ukuhlushwa kwezidakamizwa kuphezulu egazini nezicubu, futhi ukugxila kwegazi okuphumelelayo kugcinwa isikhathi eside. I-metabolite esebenzayo ye-desfuroylceftiofur ingakhiqizwa emzimbeni, futhi iphinde igaywe ibe yimikhiqizo engasebenzi ekhishwa emchameni nasendle.
ama-antibiotic e-β-lactam. Isetshenziselwa ikakhulukazi ukwelapha izifo ezibangelwa amagciwane emfuyo nezinkukhu. Okufana nengulube yebhaktheriya yokuphefumula ukutheleleka kanye nenkukhu escherichia coli, ukutheleleka kwe-salmonella.
I-Ceftiofur isetshenziswa. Umjovo we-Intramuscular: Umthamo owodwa, 1.1- 2.2mg nge-1kg isisindo somzimba wezinkomo, 3-5mg wezimvu nezingulube, 5mg wenkukhu kanye nedada, kanye ngosuku izinsuku ezintathu.
Umjovo ongaphansi kwesikhumba: amatshwele anosuku olu-1 ubudala, 0.1mg uphaphe ngalunye.
(1) Kungase kubangele ukuphazamiseka kwezitshalo emathunjini noma ukutheleleka kabili.
(2) Kukhona i-nephrotoxicity ethile.
(3) Ubuhlungu besikhashana bendawo bungenzeka.
(1)Sebenzisa manje.
(2) Umthamo kufanele ulungiswe ezilwaneni ezinokwehluleka kwezinso.
(3)Abantu abazwela kakhulu kuma-antibiotic e-beta-lactam kufanele bagweme ukuthintana nalo mkhiqizo futhi bagweme ukuchayeka ezinganeni.